What are aromatase inhibitors?What are aromatase inhibitors?

We will not rush right off the bat, but rather talk about everything in order, starting, as usual, with theory. So, aromatase inhibitors, also known as blockers or blockers, are a class of effective drugs used in medicine for the treatment of cancers, in particular breast cancer (not only).

In sports, for example, in bodybuilding, aromatase blockers are primarily useful in the course of a course of steroids, helping to reduce the concentration of estrogens, increase the level of endogenous testosterone and gonadotropic hormones. aromatase inhibitors They are usually used by athletes to prevent and / or eliminate estrogenic side effects such as gynecomastia (enlargement of the breast that occurs in men).

In more detail, in bodybuilding, aromatase inhibitors are most often used during the course of anabolic steroids for the following purposes:

Prevention and elimination of estrogenic side effects (gynecomastia, etc.);
An increase in the level of anabolic hormones in the blood (testosterone), etc.

It is important to note that aromatase inhibitors are antiestrogens by class. As many people know, testosterone in our body can be converted (converted) into estradiol. This happens with the assistance of an enzyme called aromatase. With the participation of the same enzyme, another conversion process occurs - androstenedione is converted into estrone. The purpose of the inhibitory agents described in this material is to prevent this type of transformation, and they do this, as the name implies, by blocking aromatase.